PKA Inhibitor Fragment (6-22) amide TFA is an inhibitor of cAMP-dependent protein kinase A (PKA), with a Ki of 2.8 nM. PKA Inhibitor Fragment (6-22) amide TFA can significantly reverse low-level morphine antinociceptive tolerance in mice.
Chalepensin, a furanocoumarin isolated from the rutaceae plant Ruta chalepensis L., is a selective CYP2A6 inhibitor. Chalepensin also inhibits human CYP1A1, CYP1A2, CYP2A13, CYP2C9, CYP2D6, CYP2E1, and CYP3A4.
Quercetin 3-gentiobioside is isolated from A. iwayomogi, AR and AGE formation inhibitor, demonstrates biological activities against Aldose reductase (AR) and the formation of advanced glycation endproducts (AGEs).
N-Benzylpalmitamide is a macamide isolated from Lepidium meyenii, acts as an inhibitor of fatty acid amide hydrolase (FAAH).
Militarine, a glycosidic compound isolated from Bletilla striata, exhibits plant growth-inhibitory activity.
Militarine, a glycosidic compound isolated from Bletilla striata, exhibits plant growth-inhibitory activity.
Amoxicillin is a broad-spectrum, semisynthetic aminopenicillin antibiotic with bactericidal activity.
Amoxicillin is a broad-spectrum, semisynthetic aminopenicillin antibiotic with bactericidal activity.
WAY-643895 is a casein kinase 1δ (CK1δ) inhibitor with >5% inhibition. It can be used in studies related to neurodegenerative diseases such as Alzheimer's disease.
WAY-643895 is a casein kinase 1δ (CK1δ) inhibitor with >5% inhibition. It can be used in studies related to neurodegenerative diseases such as Alzheimer's disease.
WAY-647766 is a potent Casein kinase 1δ inhibitor for Alzheimer's disease related studies.