ASTX660 is a potent, non-peptidomimetic antagonist of cIAP1/2 and XIAP, it potently inhibited the interactions between a SMAC-derived peptide and the BIR3 domains of XIAP (BIR3-XIAP) and cIAP1 (BIR3-cIAP1) with IC50 values less than 40 and 12 nmol/L, respectively.
α-Naphthoflavone is a potent and competitive aromatase inhibitor with an IC50 and a Ki of 0.5 and 0.2 μM, respectively. Alpha-Naphthoflavone can inhibit cell proliferation and induce apoptosis.
α-Naphthoflavone is a potent and competitive aromatase inhibitor with an IC50 and a Ki of 0.5 and 0.2 μM, respectively. Alpha-Naphthoflavone can inhibit cell proliferation and induce apoptosis.
Inosine (Inosine) is an endogenous purine nucleoside produced by the catabolism of adenosine. It has immunomodulatory, neuroprotective effects.
Efinaconazole (KP-103) is a triazole antifungal, it also acts as a 14α-demethylase inhibitor.
Seractide; ACTH (1-39), human is a member of the melanocortin family, stimulates production of CS by the adrenals, acts as a melanocortin receptor agonist.
Chlorotoxin is a 36 amino-acid peptide with anticancer activity, it is also a chloride channel blocker.
1-Thioglycerol, a derivatization reagent, is used to study the pH-sensitive photoluminescence of aqueous thiol-capped CdTe nanocrystals.
Seractide; ACTH (1-39), human is a member of the melanocortin family, stimulates production of CS by the adrenals, acts as a melanocortin receptor agonist.
BMS-1166 is a potent PD-1/PD-L1 interaction inhibitor, which binds to human PD-L1 and blocks its interaction with PD-1.
BMS-1166 is a potent PD-1/PD-L1 interaction inhibitor, which binds to human PD-L1 and blocks its interaction with PD-1.
Cycloleucine is antagonist of NMDA receptor associated glycine receptor, with a Ki of 600 μM. Cycloleucine is a specific inhibitor of S-adenosyl-methionine mediated methylation.